遇见数据集

LSD1-CoREST in complex with T105

收藏
Protein Data Bank Japan2025-06-25 更新2026-05-23 收录
数据链接:
官方服务:

资源简介:

LSD1-CoREST in complex with T105 Descriptor: 3-[(1R,2S)-2-(cyclobutylamino)cyclopropyl]-N-(5-methyl-1,3,4-thiadiazol-2-yl)benzamide, Lysine-specific histone demethylase 1A, REST corepressor 1, ... Authors: Caroli, J, Mattevi, A. Deposit date: 2022-11-17 Release date: 2024-06-12 Last modified: 2025-06-25 Method: X-RAY DIFFRACTION (2.91 Å) Cite: Covalent adduct Grob fragmentation underlies LSD1 demethylase-specific inhibitor mechanism of action and resistance. Nat Commun, 16, 2025

创建时间:
2022-11-17
二维码
社区交流群
二维码
科研交流群
商业服务