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PAD2 with an inhibitor

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Protein Data Bank Japan2025-09-03 更新2026-05-23 收录
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PAD2 with an inhibitor Descriptor: (2S)-2-amino-2-(1-{(5M)-5-[3,5-dichloro-6-(1-methyl-1H-pyrazol-3-yl)pyridin-2-yl]isoquinolin-1-yl}piperidin-4-yl)-N-methylacetamide, CALCIUM ION, Protein-arginine deiminase type-2 Authors: Yamaguchi, M. Deposit date: 2025-05-30 Release date: 2025-07-30 Last modified: 2025-09-03 Method: X-RAY DIFFRACTION (2.175 Å) Cite: Peptidylarginine Deiminase (PAD) Inhibitor Optimization through Displacement of a Trapped Water Molecule. Acs Med.Chem.Lett., 16, 2025

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2025-05-30
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