C-TERMINAL BROMODOMAIN OF HUMAN BRD2 WITH GSK973
收藏Protein Data Bank Japan2024-05-01 更新2026-03-21 收录
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https://pdbj.org/mine/summary/6z8p
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C-TERMINAL BROMODOMAIN OF HUMAN BRD2 WITH GSK973 Descriptor: (2~{S},3~{S})-2-(fluoranylmethyl)-~{N}7-methyl-~{N}5-[(1~{R},5~{S})-3-oxabicyclo[3.1.0]hexan-6-yl]-3-phenyl-2,3-dihydro-1-benzofuran-5,7-dicarboxamide, 1,2-ETHANEDIOL, 2-(2-{2-[2-(2-METHOXY-ETHOXY)-ETHOXY]-ETHOXY}-ETHOXY)-ETHANOL, ... Authors: Chung, C. Deposit date: 2020-06-02 Release date: 2020-10-21 Last modified: 2024-05-01 Method: X-RAY DIFFRACTION (1.55 Å) Cite: GSK973 Is an Inhibitor of the Second Bromodomains (BD2s) of the Bromodomain and Extra-Terminal (BET) Family. Acs Med.Chem.Lett., 11, 2020
创建时间:
2020-06-02



