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USP7 in complex with a novel inhibitor

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Protein Data Bank Japan2023-11-29 更新2026-03-21 收录
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USP7 in complex with a novel inhibitor Descriptor: Ubiquitin carboxyl-terminal hydrolase 7, methyl 4-[[4-[[3-[4-(aminomethyl)phenyl]-2-methyl-7-oxidanylidene-pyrazolo[4,3-d]pyrimidin-6-yl]methyl]-4-oxidanyl-piperidin-1-yl]methyl]-3-chloranyl-benzoate Authors: Liu, S.J, Zhou, X.Y, Li, M.L, Sun, H.B, Wen, X.A. Deposit date: 2020-02-26 Release date: 2021-03-10 Last modified: 2023-11-29 Method: X-RAY DIFFRACTION (2.255 Å) Cite: N-benzylpiperidinol derivatives as novel USP7 inhibitors: Structure-activity relationships and X-ray crystallographic studies. Eur.J.Med.Chem., 199, 2020
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2020-02-26
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