five

Crystal Structure Analysis of the BRD4

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Protein Data Bank Japan2024-03-27 更新2026-03-21 收录
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Crystal Structure Analysis of the BRD4 Descriptor: (2R)-2-(cyclopropylmethyl)-7-(3,5-dimethyl-1,2-oxazol-4-yl)-4H-1,4-benzoxazin-3-one, 1,2-ETHANEDIOL, Bromodomain-containing protein 4, ... Authors: Xue, X, Zhang, Y, Wang, C, Song, M. Deposit date: 2017-11-08 Release date: 2018-11-28 Last modified: 2024-03-27 Method: X-RAY DIFFRACTION (1.82 Å) Cite: Benzoxazinone-containing 3,5-dimethylisoxazole derivatives as BET bromodomain inhibitors for treatment of castration-resistant prostate cancer. Eur.J.Med.Chem., 152, 2018
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2017-11-08
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