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Co-complex CYP46A1 with 9129 (1b)

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Protein Data Bank Japan2023-10-18 更新2026-04-19 收录
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https://pdbj.org/mine/summary/7ls4
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资源简介:
Co-complex CYP46A1 with 9129 (1b) Descriptor: Cholesterol 24-hydroxylase, PROTOPORPHYRIN IX CONTAINING FE, [5,5-dimethyl-3-(2-methylphenyl)-4~{H}-pyrazol-1-yl]-pyridin-4-yl-methanone Authors: Lane, W, Yano, J. Deposit date: 2021-02-17 Release date: 2021-08-25 Last modified: 2023-10-18 Method: X-RAY DIFFRACTION (2.05 Å) Cite: Discovery of Soticlestat, a Potent and Selective Inhibitor for Cholesterol 24-Hydroxylase (CH24H). J.Med.Chem., 64, 2021
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2021-02-17
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