Crystal structure of PDE10a with a novel Imidazo[4,5-b]pyridine inhibitor
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Crystal structure of PDE10a with a novel Imidazo[4,5-b]pyridine inhibitor Descriptor: GLYCEROL, N-[cis-3-(2-methoxy-3H-imidazo[4,5-b]pyridin-3-yl)cyclobutyl]-1,3-benzothiazol-2-amine, N-[trans-3-(2-methoxy-3H-imidazo[4,5-b]pyridin-3-yl)cyclobutyl]-1,3-benzothiazol-2-amine, ... Authors: Chmait, S. Deposit date: 2014-02-21 Release date: 2014-10-01 Last modified: 2024-10-23 Method: X-RAY DIFFRACTION (2.08 Å) Cite: Discovery of Novel Imidazo[4,5-b]pyridines as Potent and Selective Inhibitors of Phosphodiesterase 10A (PDE10A). Acs Med.Chem.Lett., 5, 2014
创建时间:
2014-02-21



