Crystal Structure of the human BRD2 BD1 bromodomain in complex with a Tetrahydroquinoline analogue
收藏Protein Data Bank Japan2023-10-11 更新2026-03-21 收录
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Crystal Structure of the human BRD2 BD1 bromodomain in complex with a Tetrahydroquinoline analogue Descriptor: 1,2-ETHANEDIOL, 4-{[(2S,4R)-1-acetyl-2-methyl-6-(1H-pyrazol-3-yl)-1,2,3,4-tetrahydroquinolin-4-yl]amino}benzonitrile, Bromodomain-containing protein 2, ... Authors: White, S.W, Yun, M. Deposit date: 2018-05-10 Release date: 2019-11-13 Last modified: 2023-10-11 Method: X-RAY DIFFRACTION (1.5 Å) Cite: Bromodomain-Selective BET Inhibitors Are Potent Antitumor Agents against MYC-Driven Pediatric Cancer. Cancer Res., 80, 2020
创建时间:
2018-05-10



