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Crystal structure of JAK2 JH1 in complex with cerdulatinib

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Protein Data Bank Japan2024-11-06 更新2026-03-28 收录
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Crystal structure of JAK2 JH1 in complex with cerdulatinib Descriptor: Cerdulatinib, Tyrosine-protein kinase JAK2 Authors: Haikarainen, T. Deposit date: 2022-12-08 Release date: 2023-12-20 Last modified: 2024-11-06 Method: X-RAY DIFFRACTION (1.5 Å) Cite: Functional and Structural Characterization of Clinical-Stage Janus Kinase 2 Inhibitors Identifies Determinants for Drug Selectivity. J.Med.Chem., 67, 2024

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2022-12-08
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