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Crystal structure of murine NF-kappaB inducing kinase (NIK) bound to benzoxepin compound 2

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Protein Data Bank Japan2024-05-08 更新2026-03-21 收录
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Crystal structure of murine NF-kappaB inducing kinase (NIK) bound to benzoxepin compound 2 Descriptor: 6,7-dihydrothieno[4,5]oxepino[1,2-~{c}]pyridine-2-carboxamide, Mitogen-activated protein kinase kinase kinase 14, SULFATE ION Authors: Smith, M.A, McEwan, P.A. Deposit date: 2016-09-08 Release date: 2017-01-11 Last modified: 2024-05-08 Method: X-RAY DIFFRACTION (2.32 Å) Cite: Structure-Based Design of Tricyclic NF-kappa B Inducing Kinase (NIK) Inhibitors That Have High Selectivity over Phosphoinositide-3-kinase (PI3K). J. Med. Chem., 60, 2017
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2016-09-08
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