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BRAFV600E Kinase Domain In Complex with Chemically Linked Vemurafenib Inhibitor VEM-3-VEM

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Protein Data Bank Japan2023-09-27 更新2026-03-21 收录
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https://pdbj.org/mine/summary/5jsm
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资源简介:
BRAFV600E Kinase Domain In Complex with Chemically Linked Vemurafenib Inhibitor VEM-3-VEM Descriptor: BENZAMIDINE, CHLORIDE ION, DIMETHYL SULFOXIDE, ... Authors: Grasso, M.J, Marmorstein, R. Deposit date: 2016-05-08 Release date: 2016-09-14 Last modified: 2023-09-27 Method: X-RAY DIFFRACTION (2.19 Å) Cite: Chemically Linked Vemurafenib Inhibitors Promote an Inactive BRAF(V600E) Conformation. Acs Chem.Biol., 11, 2016
创建时间:
2016-05-08
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