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Crystal structure of RabGGTase(DELTA LRR; DELTA IG) in Complex with BMS-analogue 14

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Protein Data Bank Japan2023-09-13 更新2026-03-21 收录
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Crystal structure of RabGGTase(DELTA LRR; DELTA IG) in Complex with BMS-analogue 14 Descriptor: 4-({(3R)-7-(5-formylfuran-2-yl)-4-[(4-methoxyphenyl)sulfonyl]-1-[(1-methyl-1H-imidazol-5-yl)methyl]-2,3,4,5-tetrahydro-1H-1,4-benzodiazepin-3-yl}methyl)phenyl benzylcarbamate, CALCIUM ION, Geranylgeranyl transferase type-2 subunit alpha, ... Authors: Guo, Z, Bon, R.S, Stigter, E.A, Waldmann, H, Alexandrov, K, Blankenfeldt, W, Goody, R.S. Deposit date: 2010-12-14 Release date: 2011-05-11 Last modified: 2023-09-13 Method: X-RAY DIFFRACTION (2 Å) Cite: Structure-Guided Development of Selective RabGGTase Inhibitors. Angew.Chem.Int.Ed.Engl., 50, 2011
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2010-12-14
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