five

BAY-707 in complex with MTH1

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Protein Data Bank Japan2024-01-17 更新2026-03-21 收录
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https://pdbj.org/mine/summary/5nhy
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BAY-707 in complex with MTH1 Descriptor: 7,8-dihydro-8-oxoguanine triphosphatase, GLYCEROL, SULFATE ION, ... Authors: Ellermann, M, Eheim, A, Giese, A, Bunse, S, Nowak-Reppel, K, Neuhaus, R, Weiske, J, Quanz, M, Glasauer, A, Meyer, H, Queisser, N, Irlbacher, H, Bader, B, Rahm, F, Viklund, J, Andersson, M, Ericsson, U, Ginman, T, Forsblom, R, Lindstrom, J, Silvander, C, Tresaugues, L, Gorjanacz, M. Deposit date: 2017-03-22 Release date: 2017-07-19 Last modified: 2024-01-17 Method: X-RAY DIFFRACTION (1.72 Å) Cite: Novel Class of Potent and Cellularly Active Inhibitors Devalidates MTH1 as Broad-Spectrum Cancer Target. ACS Chem. Biol., 12, 2017
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2017-03-22
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