EGFR kinase domain mutant "TMLR" with compound 33
收藏Protein Data Bank Japan2024-03-06 更新2026-03-21 收录
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https://pdbj.org/mine/summary/5caq
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资源简介:
EGFR kinase domain mutant "TMLR" with compound 33 Descriptor: Epidermal growth factor receptor, N-[2-[(3R,4S)-3-fluoranyl-4-methoxy-piperidin-1-yl]pyrimidin-4-yl]-2-methyl-1-propan-2-yl-imidazo[4,5-c]pyridin-6-amine, SULFATE ION Authors: Eigenbrot, C, Yu, C. Deposit date: 2015-06-29 Release date: 2015-10-28 Last modified: 2024-03-06 Method: X-RAY DIFFRACTION (2.5 Å) Cite: Noncovalent Mutant Selective Epidermal Growth Factor Receptor Inhibitors: A Lead Optimization Case Study. J.Med.Chem., 58, 2015
创建时间:
2015-06-29



