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CRYSTAL STRUCTURE OF THE VEGFR2 KINASE DOMAIN IN COMPLEX WITH AXITINIB (AG-013736) (N-Methyl-2-(3-((E)-2-pyridin-2-yl-vinyl)-1H- indazol-6-ylsulfanyl)-benzamide)

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Protein Data Bank Japan2024-08-07 更新2026-03-21 收录
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https://pdbj.org/mine/summary/4ag8
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CRYSTAL STRUCTURE OF THE VEGFR2 KINASE DOMAIN IN COMPLEX WITH AXITINIB (AG-013736) (N-Methyl-2-(3-((E)-2-pyridin-2-yl-vinyl)-1H- indazol-6-ylsulfanyl)-benzamide) Descriptor: AXITINIB, VASCULAR ENDOTHELIAL GROWTH FACTOR RECEPTOR 2 Authors: McTigue, M, Wickersham, J, Pinko, C, Kania, R.S, Bender, S. Deposit date: 2012-01-24 Release date: 2012-09-26 Last modified: 2024-08-07 Method: X-RAY DIFFRACTION (1.95 Å) Cite: Molecular Conformations, Interactions, and Properties Associated with Drug Efficiency and Clinical Performance Among Vegfr Tk Inhibitors. Proc.Natl.Acad.Sci.USA, 109, 2012
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2012-01-24
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