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Co-crystal structure of PERK with compound 11

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Protein Data Bank Japan2023-10-25 更新2026-04-19 收录
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Co-crystal structure of PERK with compound 11 Descriptor: (2R)-N-[(4M)-4-(4-amino-7-methyl-7H-pyrrolo[2,3-d]pyrimidin-5-yl)-3-methylphenyl]-2-(3-fluorophenyl)-2-hydroxyacetamide, Eukaryotic translation initiation factor 2-alpha kinase 3 Authors: Zhu, G, Surman, M.D, Mulvihill, M.J. Deposit date: 2022-10-07 Release date: 2022-11-30 Last modified: 2023-10-25 Method: X-RAY DIFFRACTION (2.86 Å) Cite: Optimization of a Novel Mandelamide-Derived Pyrrolopyrimidine Series of PERK Inhibitors. Pharmaceutics, 14, 2022
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2022-10-07
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