Glucocorticoid Receptor LBD bound to GSK866

Glucocorticoid Receptor LBD bound to GSK866 Descriptor: 5-amino-N-[(2S)-2-({[(2,6-dichlorophenyl)carbonyl](ethyl)amino}methyl)-3,3,3-trifluoro-2-hydroxypropyl]-1-(4-fluorophenyl)-1H-pyrazole-4-carboxamide, GLYCEROL, Glucocorticoid receptor, ... Authors: Madauss, K.P, Williams, S.P, Mclay, I, Stewart, E.L, Bledsoe, R.K. Deposit date: 2008-08-18 Release date: 2008-11-25 Last modified: 2024-04-03 Method: X-RAY DIFFRACTION (2.15 Å) Cite: The first X-ray crystal structure of the glucocorticoid receptor bound to a non-steroidal agonist. Bioorg.Med.Chem.Lett., 18, 2008