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Crystal Structure of BAZ2B bromodomain in complex with acetylindole compound UZH50

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Protein Data Bank Japan2024-01-10 更新2026-03-21 收录
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Crystal Structure of BAZ2B bromodomain in complex with acetylindole compound UZH50 Descriptor: Bromodomain adjacent to zinc finger domain protein 2B, N-(1-acetyl-1H-indol-3-yl)-N-(5-hydroxy-2-methylphenyl)-3-(trifluoromethyl)benzamide Authors: Lolli, G, Spiliotopoulos, D, Dolbois, A, Nevado, C, Caflisch, A. Deposit date: 2015-10-11 Release date: 2015-10-21 Last modified: 2024-01-10 Method: X-RAY DIFFRACTION (1.783 Å) Cite: The "Gatekeeper" Residue Influences the Mode of Binding of Acetyl Indoles to Bromodomains. J. Med. Chem., 59, 2016

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2015-10-11
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