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Mcl-1 complexed with small molecules

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Protein Data Bank Japan2024-03-06 更新2026-03-21 收录
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Mcl-1 complexed with small molecules Descriptor: 1-[3-(naphthalen-1-yloxy)propyl]-5,6-dihydro-4H-pyrrolo[3,2,1-ij]quinoline-2-carboxylic acid, Induced myeloid leukemia cell differentiation protein Mcl-1 Authors: Zhao, B. Deposit date: 2015-04-14 Release date: 2015-04-29 Last modified: 2024-03-06 Method: X-RAY DIFFRACTION (2.5 Å) Cite: Discovery of tricyclic indoles that potently inhibit mcl-1 using fragment-based methods and structure-based design. J.Med.Chem., 58, 2015

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2015-04-14
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