C-TERMINAL BROMODOMAIN OF HUMAN BRD2 WITH (S)-N-ethyl-3-(1-methyl-1H-1,2,3-triazol-4-yl)-4-(1-phenylethoxy)benzamide
收藏Protein Data Bank Japan2024-06-19 更新2026-03-21 收录
下载链接:
https://pdbj.org/mine/summary/7nq7
下载链接
链接失效反馈官方服务:
资源简介:
C-TERMINAL BROMODOMAIN OF HUMAN BRD2 WITH (S)-N-ethyl-3-(1-methyl-1H-1,2,3-triazol-4-yl)-4-(1-phenylethoxy)benzamide Descriptor: 1,2-ETHANEDIOL, Bromodomain-containing protein 2, ~{N}-ethyl-3-(1-methyl-1,2,3-triazol-4-yl)-4-[(1~{S})-1-phenylethoxy]benzamide Authors: Chung, C. Deposit date: 2021-03-01 Release date: 2021-03-24 Last modified: 2024-06-19 Method: X-RAY DIFFRACTION (1.7 Å) Cite: Template-Hopping Approach Leads to Potent, Selective, and Highly Soluble Bromo and Extraterminal Domain (BET) Second Bromodomain (BD2) Inhibitors. J.Med.Chem., 64, 2021
创建时间:
2021-03-01



