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ROR(gamma)t ligand binding domain in complex with allosteric ligand FM26

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Protein Data Bank Japan2024-01-24 更新2026-03-21 收录
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https://pdbj.org/mine/summary/6sal
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资源简介:
ROR(gamma)t ligand binding domain in complex with allosteric ligand FM26 Descriptor: 4-[(~{E})-[3-[2-chloranyl-6-(trifluoromethyl)phenyl]-5-(1~{H}-pyrrol-3-yl)-1,2-oxazol-4-yl]methylideneamino]benzoic acid, Nuclear receptor ROR-gamma Authors: de Vries, R.M.J.M, Meijer, F.A, Doveston, R.G, Brunsveld, L. Deposit date: 2019-07-17 Release date: 2019-12-25 Last modified: 2024-01-24 Method: X-RAY DIFFRACTION (1.61 Å) Cite: Ligand-Based Design of Allosteric Retinoic Acid Receptor-Related Orphan Receptor gamma t (ROR gamma t) Inverse Agonists. J.Med.Chem., 63, 2020
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2019-07-17
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