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Crystal structure of BRD4 bromodomain 1 (BD1) in complex with C239-0012

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Protein Data Bank Japan2023-11-29 更新2026-04-19 收录
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Crystal structure of BRD4 bromodomain 1 (BD1) in complex with C239-0012 Descriptor: 3-methyl-6-(4-methylpiperidin-1-yl)-[1,2,4]triazolo[4,3-b]pyridazine, Bromodomain-containing protein 4, FORMIC ACID, ... Authors: Park, T.H, Lee, B.I. Deposit date: 2022-08-27 Release date: 2023-01-18 Last modified: 2023-11-29 Method: X-RAY DIFFRACTION (1.528 Å) Cite: Crystal structure of [1,2,4]triazolo[4,3-b]pyridazine derivatives as BRD4 bromodomain inhibitors and structure-activity relationship study. Sci Rep, 13, 2023
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