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Crystal structure of TYK2 in complex with peficitinib

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Protein Data Bank Japan2024-03-27 更新2026-03-21 收录
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Crystal structure of TYK2 in complex with peficitinib Descriptor: 4-[[(1S,3R)-5-oxidanyl-2-adamantyl]amino]-1H-pyrrolo[2,3-b]pyridine-5-carboxamide, Non-receptor tyrosine-protein kinase TYK2 Authors: Nomura, N, Tomimoto, Y. Deposit date: 2018-07-18 Release date: 2018-08-15 Last modified: 2024-03-27 Method: X-RAY DIFFRACTION (1.98 Å) Cite: Discovery and structural characterization of peficitinib (ASP015K) as a novel and potent JAK inhibitor Bioorg. Med. Chem., 26, 2018

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2018-07-18
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