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Crystal structure of CYP3A4 bound to an inhibitor

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Protein Data Bank Japan2026-08-12 更新2026-05-23 收录
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Crystal structure of CYP3A4 bound to an inhibitor Descriptor: Cytochrome P450 3A4, PROTOPORPHYRIN IX CONTAINING FE, {N-[([2,2'-bipyridin]-5-yl-kappa~2~N~1~,N~1'~)methyl]-3-(pyridin-4-yl)propanamide}bis[2-(quinolin-2-yl-kappaN)-1-benzothiophen-3-yl-kappaC~3~]iridium(1+) Authors: Sevrioukova, I.F. Deposit date: 2022-10-24 Release date: 2023-02-01 Last modified: 2026-08-12 Method: X-RAY DIFFRACTION (2.15 Å) Cite: Dynamic Ir(III) Photosensors for the Major Human Drug-Metabolizing Enzyme Cytochrome P450 3A4. Inorg.Chem., 62, 2023

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2022-10-24
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