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TBK1 in complex with inhibitor compound 24

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Protein Data Bank Japan2024-05-15 更新2026-03-21 收录
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TBK1 in complex with inhibitor compound 24 Descriptor: 1-[4-[(1~{R})-1-[2-[[5-[1-(cyclopropylmethyl)pyrazol-4-yl]-1~{H}-benzimidazol-2-yl]amino]pyridin-4-yl]ethyl]piperazin-1-yl]-3,3,3-tris(fluoranyl)propan-1-one, Serine/threonine-protein kinase TBK1 Authors: Panne, D, Hillig, R.C, Rengachari, S. Deposit date: 2019-05-22 Release date: 2020-01-01 Last modified: 2024-05-15 Method: X-RAY DIFFRACTION (3.29 Å) Cite: Discovery of BAY-985, a Highly Selective TBK1/IKK epsilon Inhibitor. J.Med.Chem., 63, 2020

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2019-05-22
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