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Human PPAR gamma ligand binding domain in complex with a gamma selective agonist mekt21

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Protein Data Bank Japan2023-11-08 更新2026-03-21 收录
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https://pdbj.org/mine/summary/3vso
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资源简介:
Human PPAR gamma ligand binding domain in complex with a gamma selective agonist mekt21 Descriptor: (2R)-2-benzyl-3-[4-propoxy-3-({[4-(pyrimidin-2-yl)benzoyl]amino}methyl)phenyl]propanoic acid, Peroxisome proliferator-activated receptor gamma Authors: Oyama, T, Waku, T, Ohashi, M, Morikawa, K, Miyachi, H. Deposit date: 2012-04-30 Release date: 2013-05-01 Last modified: 2023-11-08 Method: X-RAY DIFFRACTION (2 Å) Cite: Design and synthesis of a series of alpha-benzyl phenylpropanoic acid-type peroxisome proliferator-activated receptor (PPAR) gamma partial agonists with improved aqueous solubility Bioorg.Med.Chem., 21, 2013
创建时间:
2012-04-30
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