five

GLK co-crystal structure with aminopyrrolopyrimidine inhibitor

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Protein Data Bank Japan2024-10-30 更新2026-03-21 收录
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GLK co-crystal structure with aminopyrrolopyrimidine inhibitor Descriptor: 5-[2-(piperidin-4-yl)-1,3-thiazol-5-yl]-3-[(pyridin-4-yl)methoxy]pyridin-2-amine, Mitogen-activated protein kinase kinase kinase kinase 3 Authors: Silvian, L.F, Marcotte, D. Deposit date: 2016-04-03 Release date: 2016-10-26 Last modified: 2024-10-30 Method: X-RAY DIFFRACTION (2.85 Å) Cite: Germinal-center kinase-like kinase co-crystal structure reveals a swapped activation loop and C-terminal extension. Protein Sci., 26, 2017
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2016-04-03
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