遇见数据集

USP7 IN COMPLEX WITH LIGAND COMPOUND 18

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Protein Data Bank Japan2024-11-13 更新2026-03-21 收录
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USP7 IN COMPLEX WITH LIGAND COMPOUND 18 Descriptor: 1-({7-[(2R)-5-chloro-2-(piperazine-1-carbonyl)-2,3-dihydro-1-benzofuran-7-yl]thieno[3,2-b]pyridin-2-yl}methyl)-1H-pyrrole-2,5-dione, ACETATE ION, Ubiquitin carboxyl-terminal hydrolase 7 Authors: Leger, P.R, Wustrow, D.J, Hu, D.X, Krapp, S, Maskos, K, Blaesse, M. Deposit date: 2020-01-29 Release date: 2020-04-29 Last modified: 2024-11-13 Method: X-RAY DIFFRACTION (2.93 Å) Cite: Discovery of Potent, Selective, and Orally Bioavailable Inhibitors of USP7 with In Vivo Antitumor Activity. J.Med.Chem., 63, 2020

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2020-01-29
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