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Crystal structure of the PPARgamma-LBD complexed with compound 13ab

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Protein Data Bank Japan2023-11-22 更新2026-03-21 收录
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Crystal structure of the PPARgamma-LBD complexed with compound 13ab Descriptor: 3-{[6-(4-chloro-3-fluorophenoxy)-1-methyl-1H-benzimidazol-2-yl]methoxy}benzoic acid, CHLORIDE ION, Peptide from Peroxisome proliferator-activated receptor gamma coactivator 1-alpha, ... Authors: Matsui, Y, Hanzawa, H. Deposit date: 2018-01-19 Release date: 2018-10-17 Last modified: 2023-11-22 Method: X-RAY DIFFRACTION (1.8 Å) Cite: Discovery of DS-6930, a potent selective PPAR gamma modulator. Part I: Lead identification. Bioorg. Med. Chem., 26, 2018

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2018-01-19
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