遇见数据集

tubulin-cryptophycin complex

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Protein Data Bank Japan2024-06-12 更新2026-04-19 收录
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tubulin-cryptophycin complex Descriptor: 2-(N-MORPHOLINO)-ETHANESULFONIC ACID, 2-[(3~{S},10~{R},13~{E},16~{S})-10-[(3-chloranyl-4-methoxy-phenyl)methyl]-6,6-dimethyl-2,5,9,12-tetrakis(oxidanylidene)-16-[(1~{S})-1-[(2~{R},3~{R})-3-phenyloxiran-2-yl]ethyl]-1,4-dioxa-8,11-diazacyclohexadec-13-en-3-yl]ethanoic acid, CALCIUM ION, ... Authors: Abel, A.C, Muehlethaler, T, Dessin, C, Steinmetz, M.O, Sewald, N, Prota, A.E. Deposit date: 2023-11-21 Release date: 2024-05-22 Last modified: 2024-06-12 Method: X-RAY DIFFRACTION (2.2 Å) Cite: Bridging the maytansine and vinca sites: Cryptophycins target beta-tubulin's T5-loop. J.Biol.Chem., 300, 2024

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2023-11-21
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