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Crystal Structure of Caspase-3 with Peptide Inhibitor Ac-VDV(DAB)D-CHO

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Protein Data Bank Japan2024-10-30 更新2026-04-19 收录
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Crystal Structure of Caspase-3 with Peptide Inhibitor Ac-VDV(DAB)D-CHO Descriptor: ACE-VAL-ASP-VAL-DAB-ASP, Caspase-3 subunit p12, Caspase-3 subunit p17 Authors: Fuller, J.L, Finzel, B.C. Deposit date: 2021-09-30 Release date: 2022-01-05 Last modified: 2024-10-30 Method: X-RAY DIFFRACTION (3.25 Å) Cite: Structure-Based Design and Biological Evaluation of Novel Caspase-2 Inhibitors Based on the Peptide AcVDVAD-CHO and the Caspase-2-Mediated Tau Cleavage Sequence YKPVD314. Acs Pharmacol Transl Sci, 5, 2022

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2021-09-30
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