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Structure of bromodomain of CREBBP with a pyrazolo[4,3-c]pyridin fragment

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Protein Data Bank Japan2024-01-17 更新2026-03-21 收录
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Structure of bromodomain of CREBBP with a pyrazolo[4,3-c]pyridin fragment Descriptor: 1,2-ETHANEDIOL, 1-(3-phenyl-1,4,6,7-tetrahydropyrazolo[4,3-c]pyridin-5-yl)propan-1-one, CREB-binding protein Authors: Filippakopoulos, P, Picaud, S, Knapp, S, von Delft, F, Bountra, C, Arrowsmith, C.H, Edwards, A, Structural Genomics Consortium (SGC) Deposit date: 2016-09-11 Release date: 2016-10-12 Last modified: 2024-01-17 Method: X-RAY DIFFRACTION (1.79 Å) Cite: Discovery of New Bromodomain Scaffolds by Biosensor Fragment Screening. ACS Med Chem Lett, 7, 2016
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2016-09-11
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