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Crystal structure of murine NF-kappaB inducing kinase (NIK) bound to Imidazobenzoxepin Compound 3

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Protein Data Bank Japan2024-05-08 更新2026-03-21 收录
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Crystal structure of murine NF-kappaB inducing kinase (NIK) bound to Imidazobenzoxepin Compound 3 Descriptor: 10-(3-methyl-3-oxidanyl-but-1-ynyl)-5,6-dihydroimidazo[1,2-d][1,4]benzoxazepine-2-carboxamide, Mitogen-activated protein kinase kinase kinase 14, SULFATE ION Authors: Smith, M.A, McEwan, P, Hymowitz, S.G. Deposit date: 2016-09-08 Release date: 2017-01-11 Last modified: 2024-05-08 Method: X-RAY DIFFRACTION (2.41 Å) Cite: Structure-Based Design of Tricyclic NF-kappa B Inducing Kinase (NIK) Inhibitors That Have High Selectivity over Phosphoinositide-3-kinase (PI3K). J. Med. Chem., 60, 2017
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2016-09-08
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