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Crystal structure of DNPH1 bound by compound 39.

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Protein Data Bank Japan2025-12-10 更新2026-04-19 收录
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Crystal structure of DNPH1 bound by compound 39. Descriptor: 3-(3-methoxyphenyl)-4-[[4-[[(3~{S})-1-pyridazin-3-ylpyrrolidin-3-yl]amino]quinazolin-2-yl]amino]benzoic acid, 5-hydroxymethyl-dUMP N-hydrolase, CHLORIDE ION, ... Authors: Collie, G.W. Deposit date: 2025-01-27 Release date: 2025-11-12 Last modified: 2025-12-10 Method: X-RAY DIFFRACTION (1.217 Å) Cite: Discovery and Optimization of a Non-Nucleoside-Based Series of Inhibitors of 2'-Deoxynucleoside 5'-Monophosphate Glycosidase (DNPH1). J.Med.Chem., 68, 2025
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2025-01-27
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