five

CDK6 (monomeric) in complex with inhibitor

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Protein Data Bank Japan2023-09-13 更新2026-03-21 收录
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CDK6 (monomeric) in complex with inhibitor Descriptor: Cyclin-dependent kinase 6, {5-[4-(dimethylamino)piperidin-1-yl]-1H-imidazo[4,5-b]pyridin-2-yl}[2-(isoquinolin-4-yl)pyridin-4-yl]methanone Authors: Chopra, R, Xu, M. Deposit date: 2012-05-02 Release date: 2013-02-06 Last modified: 2023-09-13 Method: X-RAY DIFFRACTION (2.7 Å) Cite: Fragment-Based Discovery of 7-Azabenzimidazoles as Potent, Highly Selective, and Orally Active CDK4/6 Inhibitors. ACS Med Chem Lett, 3, 2012
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2012-05-02
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