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Trypanosoma brucei PTR1 in complex with inhibitor WH16

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Protein Data Bank Japan2025-10-01 更新2026-03-21 收录
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Trypanosoma brucei PTR1 in complex with inhibitor WH16 Descriptor: (2R,3S)-1,4-DIMERCAPTOBUTANE-2,3-DIOL, (2S,3S)-1,4-DIMERCAPTOBUTANE-2,3-DIOL, 2,3-DIHYDROXY-1,4-DITHIOBUTANE, ... Authors: Nerini, E, Dawson, A, Hunter, W.N, Costi, M.P. Deposit date: 2011-05-03 Release date: 2012-05-23 Last modified: 2025-10-01 Method: X-RAY DIFFRACTION (1.8 Å) Cite: Exploiting the 2-Amino-1,3,4-thiadiazole Scaffold To Inhibit Trypanosoma brucei Pteridine Reductase in Support of Early-Stage Drug Discovery. ACS Omega, 2, 2017
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2011-05-03
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