JAK2 Pseudokinase V617F in complex with AT9283
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JAK2 Pseudokinase V617F in complex with AT9283 Descriptor: 1-cyclopropyl-3-{3-[5-(morpholin-4-ylmethyl)-1H-benzimidazol-2-yl]-1H-pyrazol-4-yl}urea, Tyrosine-protein kinase Authors: Li, Q, Li, K, Eck, M.J. Deposit date: 2018-04-13 Release date: 2019-03-20 Last modified: 2024-10-30 Method: X-RAY DIFFRACTION (3.192 Å) Cite: Discovery and Structural Characterization of ATP-Site Ligands for the Wild-Type and V617F Mutant JAK2 Pseudokinase Domain. ACS Chem. Biol., 14, 2019
创建时间:
2018-04-13



