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X-ray structure of LFA-1 I-domain in complex with LFA703 at 2.2A resolution

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Protein Data Bank Japan2023-10-25 更新2026-03-21 收录
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X-ray structure of LFA-1 I-domain in complex with LFA703 at 2.2A resolution Descriptor: 8-[2-((2S)-4-HYDROXY-1-{[5-(HYDROXYMETHYL)-6-METHOXY-2-NAPHTHYL]METHYL}-6-OXOPIPERIDIN-2-YL)ETHYL]-3,7-DIMETHYL-1,2,3,7,8,8A-HEXAHYDRONAPHTHALEN-1-YL 2-METHYLBUTANOATE, Integrin alpha-L, MAGNESIUM ION Authors: Weitz-Schmidt, G, Welzenbach, K, Dawson, J, Kallen, J. Deposit date: 2004-09-06 Release date: 2004-09-21 Last modified: 2023-10-25 Method: X-RAY DIFFRACTION (2.2 Å) Cite: Improved lymphocyte function-associated antigen-1 (LFA-1) inhibition by statin derivatives: molecular basis determined by x-ray analysis and monitoring of LFA-1 conformational changes in vitro and ex vivo J.Biol.Chem., 279, 2004
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2004-09-06
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