Notum_ARUK3001185
收藏Protein Data Bank Japan2024-11-20 更新2026-04-19 收录
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https://pdbj.org/mine/summary/7pk3
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Notum_ARUK3001185 Descriptor: 1-[2,4-bis(chloranyl)-3-(trifluoromethyl)phenyl]-1,2,3-triazole, 2-acetamido-2-deoxy-beta-D-glucopyranose, DIMETHYL SULFOXIDE, ... Authors: Vecchia, L, Hillier, J, Zhao, Y, Fish, P, Jones, E.Y. Deposit date: 2021-08-25 Release date: 2022-09-07 Last modified: 2024-11-20 Method: X-RAY DIFFRACTION (1.41 Å) Cite: Design of a Potent, Selective, and Brain-Penetrant Inhibitor of Wnt-Deactivating Enzyme Notum by Optimization of a Crystallographic Fragment Hit. J.Med.Chem., 65, 2022
创建时间:
2021-08-25



