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Complex of PI3K gamma with an inhibitor

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Protein Data Bank Japan2023-11-01 更新2026-03-21 收录
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Complex of PI3K gamma with an inhibitor Descriptor: 1-methyl-3-naphthalen-2-yl-1H-pyrazolo[3,4-d]pyrimidin-4-amine, Phosphatidylinositol-4,5-bisphosphate 3-kinase catalytic subunit gamma isoform Authors: Apsel, B, Blair, J.A, Gonzalez, B.Z, Nazif, T.M, Feldman, M.E, Williams, R.L, Shokat, K.M, Knight, Z.A. Deposit date: 2008-09-25 Release date: 2008-10-14 Last modified: 2023-11-01 Method: X-RAY DIFFRACTION (2.4 Å) Cite: Targeted polypharmacology: discovery of dual inhibitors of tyrosine and phosphoinositide kinases Nat.Chem.Biol., 4, 2008
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2008-09-25
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