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Aurora-A Inhibitor Structure

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Protein Data Bank Japan2024-11-06 更新2026-03-21 收录
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Aurora-A Inhibitor Structure Descriptor: 1,2-ETHANEDIOL, 4-{[9-CHLORO-7-(2,6-DIFLUOROPHENYL)-5H-PYRIMIDO[5,4-D][2]BENZAZEPIN-2-YL]AMINO}BENZOIC ACID, ACETATE ION, ... Authors: Kosmopoulou, M, Bayliss, R. Deposit date: 2009-09-22 Release date: 2010-01-26 Last modified: 2024-11-06 Method: X-RAY DIFFRACTION (2.4 Å) Cite: Crystal Structure of an Aurora-A Mutant that Mimics Aurora-B Bound to Mln8054: Insights Into Selectivity and Drug Design. Biochem.J., 427, 2010
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2009-09-22
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