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Bovine GRK2 in complex with Gbetagamma subunits and CCG215022

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Protein Data Bank Japan2023-09-27 更新2026-03-21 收录
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Bovine GRK2 in complex with Gbetagamma subunits and CCG215022 Descriptor: (4S)-4-{4-fluoro-3-[(pyridin-2-ylmethyl)carbamoyl]phenyl}-N-(1H-indazol-5-yl)-6-methyl-2-oxo-1,2,3,4-tetrahydropyrimidine-5-carboxamide, Beta-adrenergic receptor kinase 1, Guanine nucleotide-binding protein G(I)/G(S)/G(O) subunit gamma-2, ... Authors: Cato, M.C, Waninger-Saroni, J, Tesmer, J.J.G. Deposit date: 2016-01-05 Release date: 2016-05-11 Last modified: 2023-09-27 Method: X-RAY DIFFRACTION (2.56 Å) Cite: Structure-Based Design, Synthesis, and Biological Evaluation of Highly Selective and Potent G Protein-Coupled Receptor Kinase 2 Inhibitors. J.Med.Chem., 59, 2016
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2016-01-05
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