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PDK1 mutant bound to allosteric disulfide fragment activator 2A2

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Protein Data Bank Japan2024-11-27 更新2026-03-21 收录
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https://pdbj.org/mine/summary/3orz
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PDK1 mutant bound to allosteric disulfide fragment activator 2A2 Descriptor: 3-(1H-INDOL-3-YL)-4-{1-[2-(1-METHYLPYRROLIDIN-2-YL)ETHYL]-1H-INDOL-3-YL}-1H-PYRROLE-2,5-DIONE, 3-phosphoinositide-dependent protein kinase 1, 4-[4-(3-chlorophenyl)piperazin-1-yl]-4-oxobutane-1-thiol Authors: Sadowsky, J.D, Wells, J.A. Deposit date: 2010-09-08 Release date: 2011-03-23 Last modified: 2024-11-27 Method: X-RAY DIFFRACTION (1.9995 Å) Cite: Turning a protein kinase on or off from a single allosteric site via disulfide trapping. Proc.Natl.Acad.Sci.USA, 108, 2011
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2010-09-08
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