five

CDK8/CyclinC in complex with drug ETP-50775

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Protein Data Bank Japan2024-01-24 更新2026-03-21 收录
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CDK8/CyclinC in complex with drug ETP-50775 Descriptor: (2~{R})-butane-1,2-diol, 1-[4-chloranyl-3-(trifluoromethyl)phenyl]-3-(5-oxidanylidene-6-pyridin-4-yl-pyrido[2,3-b][1,5]benzoxazepin-9-yl)urea, Cyclin-C, ... Authors: Munoz, I.G, Pastor, J, Martinez, S. Deposit date: 2019-12-12 Release date: 2020-11-18 Last modified: 2024-01-24 Method: X-RAY DIFFRACTION (2.8 Å) Cite: Pyrido[2,3-b][1,5]benzoxazepin-5(6H)-one derivatives as CDK8 inhibitors. Eur.J.Med.Chem., 201, 2020
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2019-12-12
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