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Human Tankyrase 1 with small molecule inhibitor

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Protein Data Bank Japan2023-12-27 更新2026-03-21 收录
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资源简介:
Human Tankyrase 1 with small molecule inhibitor Descriptor: 2-(4-{6-[(3S)-3,4-dimethylpiperazin-1-yl]-4-methylpyridin-3-yl}phenyl)-8-(hydroxymethyl)quinazolin-4(3H)-one, Tankyrase-1, ZINC ION Authors: Kazmirski, S.L, Johannes, J, Boriack-Sjodin, P.A, Howard, T. Deposit date: 2014-08-20 Release date: 2015-05-13 Last modified: 2023-12-27 Method: X-RAY DIFFRACTION (1.95 Å) Cite: Pyrimidinone nicotinamide mimetics as selective tankyrase and wnt pathway inhibitors suitable for in vivo pharmacology. Acs Med.Chem.Lett., 6, 2015
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2014-08-20
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