Crystal structure of SARS-CoV-2 Mpro in complex with RK-54
收藏Protein Data Bank Japan2025-02-26 更新2026-04-19 收录
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Crystal structure of SARS-CoV-2 Mpro in complex with RK-54 Descriptor: (2R,3R)-3-[[(2S)-3-cyclopropyl-2-[3-(2-methylpropanoylamino)-2-oxidanylidene-pyridin-1-yl]propanoyl]amino]-N-methyl-2-oxidanyl-4-[(3S)-2-oxidanylidenepyrrolidin-3-yl]butanamide, 3C-like proteinase nsp5 Authors: El kilani, H, Hilgenfeld, R. Deposit date: 2024-04-25 Release date: 2025-01-29 Last modified: 2025-02-26 Method: X-RAY DIFFRACTION (2.45 Å) Cite: Structure-Based Optimization of Pyridone alpha-Ketoamides as Inhibitors of the SARS-CoV-2 Main Protease. J.Med.Chem., 68, 2025
创建时间:
2024-04-25



