Tris(pentafluorophenyl)borane-Catalyzed Stereoselective <i>C</i>‑Glycosylation of Indoles with Glycosyl Trichloroacetimidates: Access to 3‑Indolyl‑<i>C</i>‑glycosides
收藏NIAID Data Ecosystem2026-03-12 收录
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An efficient and highly regioselective method for the synthesis of 3-indolyl-C-glycosides has been developed through coupling of glycosyl trichloroacetimidates with a wide range of substituted indoles in the presence of catalytic amounts of B(C6F5)3 within a few minutes. This methodology has a wide scope of substrates under mild reaction conditions and provides exclusively β-stereoselective 3-indolyl-C-glycosides in 64–87% yields.
创建时间：
2021-05-31
