ERK5 in complex with Pyrrole Carboxamide scaffold
收藏Protein Data Bank Japan2024-01-31 更新2026-04-19 收录
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https://pdbj.org/mine/summary/7pus
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ERK5 in complex with Pyrrole Carboxamide scaffold Descriptor: 4-[3,6-bis(chloranyl)-2-fluoranyl-phenyl]carbonyl-~{N}-(1-methylpyrazol-4-yl)-1~{H}-pyrrole-2-carboxamide, Mitogen-activated protein kinase 7 Authors: Tucker, J.A, Martin, M.P, Endicott, J.A, Noble, M.E.N. Deposit date: 2021-09-30 Release date: 2022-05-11 Last modified: 2024-01-31 Method: X-RAY DIFFRACTION (2.59 Å) Cite: Parallel Optimization of Potency and Pharmacokinetics Leading to the Discovery of a Pyrrole Carboxamide ERK5 Kinase Domain Inhibitor. J.Med.Chem., 65, 2022
创建时间:
2021-09-30



