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huCaspase-6 in complex with inhibitor 3a

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Protein Data Bank Japan2024-10-16 更新2026-05-23 收录
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huCaspase-6 in complex with inhibitor 3a Descriptor: (3R,5S)-1-(ethanesulfonyl)-5-phenyl-N-[4-(trifluoromethoxy)phenyl]piperidine-3-carboxamide (bound form), 1,2-ETHANEDIOL, Caspase-6 subunit p11, ... Authors: Zhao, Y, Fan, P, Liu, J, Wang, Y, Van Horn, K, Wang, D, Medina-Cleghorn, D, Lee, P, Bryant, C, Altobelli, C, Jaishankar, P, Ng, R.A, Ambrose, A.J, Tang, Y, Arkin, M.R, Renslo, A.R. Deposit date: 2022-09-11 Release date: 2023-05-10 Last modified: 2024-10-16 Method: X-RAY DIFFRACTION (2.14 Å) Cite: Engaging a Non-catalytic Cysteine Residue Drives Potent and Selective Inhibition of Caspase-6. J.Am.Chem.Soc., 145, 2023

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2022-09-11
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