Human cGAS catalytic domain bound with XL-3156
收藏Protein Data Bank Japan2025-09-10 更新2026-04-19 收录
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Human cGAS catalytic domain bound with XL-3156 Descriptor: 2-(1~{H}-benzimidazol-2-yl)-4-[[1-(1~{H}-benzimidazol-2-yl)-3-methyl-5-oxidanyl-pyrazol-4-yl]-pyridin-2-yl-methyl]-5-methyl-pyrazol-3-ol, Cyclic GMP-AMP synthase, ZINC ION Authors: Zhao, W.F, Li, M.J, Xu, Y.C. Deposit date: 2024-08-07 Release date: 2025-06-04 Last modified: 2025-09-10 Method: X-RAY DIFFRACTION (2.2 Å) Cite: De novo design of protein condensation inhibitors by targeting an allosteric site of cGAS. Nat Commun, 16, 2025
创建时间:
2024-08-07



